Buy Varenicline tartrate | | Chantix | Champix | HSDB7591 | CP526555|375815-87-5|Signal Transduction |from supplier chembestbuy.com|Research only

Home

Add Favorites

Search Product

Live Chat

E-mail

Pharmacology

Inhibitors

Receptors

Hedgehog Signaling Pathway

Research Area

Cardiovascular System

Product Type

Vitamin D series compounds

Toxins

　 More +

Browse Alphabetically by Name

ALL	A	B	C	D	E	F
G	H	I	J	K	L	M
N	O	P	Q	R	S	T
U	V	W	X	Y	Z	Others

Catalog No.:	CL2240
CAS No.:	375815-87-5
Synonym:	CP 526555-18; Champix tartrate; Chantix tartrate
Chemical Name:	(6R,10S)-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g]quinoxaline (2R,3R)-2,3-dihydroxysuccinate
Molecular Formula:	C₁₇H₁₉N₃O₆
Molecular Weight:	361.37

Technical Data:

Appearance:	White powder
Solubility:	Soluble in water
Purity:	>99%
Storage:	Store at room temperature
Original QC Data:
Shipping Conditions:	Ambient Temp.

Size	Price	Stock
20 mg	USD 136	In stock
50 mg	USD 188	In stock
100 mg	USD 266	In stock

Biological Activity:

Orally active, subtype-selective partial agonist at α4β2 nicotinic receptors (K_i values are 0.06, 240, 322 and 3540 nM for α4β2, α3β4, α7, α1βγδ receptors respectively). Reduces nicotine-evoked dopamine release in vitro and decreases nicotine self-administration in vivo.

References:

Coe JW et al. Varenicline: an alpha4beta2 nicotinic receptor partial agonist for smoking cessation. J Med Chem 48:3474-7 (2005).

View Related Products by Target:

Cyclopamine(11-Deoxyjervine)

(+)-Egenine