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C14761 Ketanserin(R 41 468) (74050-98-9)

Catalog No.:	C14761
CAS No.:	74050-98-9
Synonym:	Ketanserin [USAN:INN:BAN]; Ketanserin; 2,4(1H,3H)-Quinazolinedione, 3-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-; 3-(2-(4-(p-Fluorobenzoyl)piperidino)ethyl)-2,4-(1H,3H)-quinazolinedione; Ketanserina; Ketanserina [INN-Spanish]; Ketanserine; Ketanserine [INN-French]; Ketanserinum; Ketanserinum [INN-Latin]; Ketaserin; R 41,468; UNII-97F9DE4CT4; 3-{2-[4-(4-fluorobenzoyl)piperidin-1-yl]ethyl}quinazoline-2,4(1H,3H)-dione
Chemical Name:	3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4[1H,3H]-quinazolinedione
Molecular Formula:	C₂₂H₂₂FN₃O₃
Molecular Weight:	395.43

Technical Data:

Appearance:	off-white power
Solubility:	soluble in DMSO
Purity:	>98%
Storage:	at -20℃ 2 years
Original QC Data:
Shipping Conditions:	Ambient Temp.

Price and Availability of Ketanserin(R 41 468):

Size	Price	Stock
10mg	USD	In stock
50mg	USD	In stock
100mg	USD	In stock

Biological Activity:

Ketanserin is a drug for 5 - HT receptor blocking, and it is selective blocking for the 5HT2 receptor, moreover, it does some weak antagonism toα and H receptor. To Hypertensive patients, Ketanserin can lower the the perivascular resistance, significant effect on Renal vascular, at the same time, it has no antihypertensive effect in normal subjects. It also be used to discriminate between 5-HT1Dand 5-HT1B receptor subtypes.

References:

Solubilized serotonin receptors from rat and dog brain. Selective labelling with [3H]ketanserin. B. Ilien et al. FEBS Lett. 138, 311, (1982).

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